Our review on selectivity of chemical probes targeting bromodomains is now published in Future Medicinal Chemistry

  • Front page
  • Figure 2. Structure and molecular recognition of BET bromodomains.
  • Figure 3.  CREBBP/EP300 bromodomain.
  • Figure 4. BRD9 bromodomain.
  • Figure 5. BAZ2B bromodomain.
  • Figure 7. BRPF and ATAD2 bromodomains.
  • Figure 8. Selectivity between BD1 and BD2 BET bromodomains.
  • Figure 9. Bump-and-hole approach.
  • Figure 10. Dual bromodomain/kinase inhibitors.

Read our open access review without restriction here.